Pharmacodynamics cefquinme yog lub cim thib plaub ntawm cephalosporin tshuaj tua kab mob rau tsiaj. Los ntawm inhibiting lub synthesis ntawm cell phab ntsa kom ua tiav cov nyhuv bactericidal, muaj ib tug dav spectrum antibacterial kev ua si, ruaj khov rau β -lactamase. Hauv vitro bacteriostatic kuaj pom tias cefquinoxime rhiab heev rau cov kab mob gram-positive thiab gram- negative. Xws li escherichia coli, citrobacter, klebsiella, pasteurella, proteus, salmonella, serratia marcescens, haemophilus bovis, actinomyces pyogenes, bacillus spp, corynebacterium, staphylococcus aureus, kab mob streptococcus, prevotella, actinobacillus thiab erysipelas suis.
Pharmacokinetic npua tau txhaj nrog 2mg ntawm cefquinoxime intraday ib 1kg ntawm lub cev qhov hnyav, thiab cov ntshav siab nce mus txog qhov siab tshaj plaws tom qab 0.4 teev, qhov siab tshaj plaws concentration yog 5.93µg / ml, tshem tawm ib nrab-lub neej yog li 1.4 teev, thiab thaj tsam hauv qab cov tshuaj nkhaus yog 12.34µgh·
β-lactam tshuaj tua kab mob yog siv los kho cov kab mob ua pa los ntawm Pasteurella multocida lossis actinobacillus pleuropneumoniae.
Kev txhaj tshuaj intramuscular: ib koob, 1mg rau 1kg lub cev hnyav, 1mg hauv nyuj, 2mg hauv yaj thiab npua, ib hnub ib zaug, rau 3-5 hnub.
Tsis muaj kev phiv tshwm sim tau raug pom raws li kev siv thiab ntau npaum li cas.
1. Tsiaj txhu yuav tsum tsis txhob siv tshuaj tua kab mob beta-lactam.
2. Tsis txhob tiv tauj cov khoom no yog tias koj ua xua rau penicillin thiab cephalosporin tshuaj tua kab mob.
3. Siv thiab sib tov tam sim no.
4. Cov khoom no yuav tsim npuas thaum yaj, thiab yuav tsum tau them sai sai rau thaum ua haujlwm.